FDA drug class

Kinase Inhibitors list

Every FDA-approved prescription drug the FDA NDC directory tags with the Kinase Inhibitor [EPC] class, with brand names and DEA schedules.

Source: FDA NDC Directory file dated 2026-10-22. Publisher page

The FDA NDC directory lists 71 single-ingredient drugs in this class: abemaciclib, acalabrutinib, afatinib, alectinib, avapritinib, axitinib, bosutinib, brigatinib, and more.

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Kinase Inhibitors (71)

Kinase Inhibitors: FDA Kinase Inhibitor class
Drug	Brand names	Type	NDC listings	DEA schedule
Abemaciclib	Verzenio	Single ingredient	4	Not controlled
Acalabrutinib	Calquence	Single ingredient	3	Not controlled
Afatinib	Gilotrif	Single ingredient	6	Not controlled
Alectinib	Alecensa	Single ingredient	1	Not controlled
Avapritinib	Ayvakit	Single ingredient	5	Not controlled
Axitinib	Inlyta	Single ingredient	4	Not controlled
Bosutinib	Bosulif	Single ingredient	11	Not controlled
Brigatinib	Alunbrig	Single ingredient	3	Not controlled
Cabozantinib s-malate	Cabometyx, Cometriq	Single ingredient	4	Not controlled
Capmatinib	Tabrecta	Single ingredient	2	Not controlled
Ceritinib	Zykadia	Single ingredient	1	Not controlled
Cobimetinib	Cotellic	Single ingredient	1	Not controlled
Crizotinib	Xalkori	Single ingredient	5	Not controlled
Dabrafenib	Tafinlar	Single ingredient	3	Not controlled
Dasatinib	Sprycel, Phyrago	Single ingredient	102	Not controlled
Erdafitinib	Balversa	Single ingredient	3	Not controlled
Erlotinib	None listed	Single ingredient	27	Not controlled
Everolimus	Afinitor, Zortress	Single ingredient	85	Not controlled
Futibatinib	Lytgobi	Single ingredient	2	Not controlled
Gedatolisib	Revtorpyk	Single ingredient	1	Not controlled
Gefitinib	Iressa	Single ingredient	5	Not controlled
Ibrutinib	Imbruvica	Single ingredient	6	Not controlled
Idelalisib	Zydelig	Single ingredient	2	Not controlled
Imatinib	Gleevec, Imkeldi	Single ingredient	45	Not controlled
Inavolisib	Itovebi	Single ingredient	2	Not controlled
Lapatinib ditosylate	Tykerb	Single ingredient	4	Not controlled
Larotrectinib	Vitrakvi	Single ingredient	7	Not controlled
Lazertinib	Lazcluze	Single ingredient	2	Not controlled
Leniolisib	Joenja	Single ingredient	3	Not controlled
Lenvatinib	Lenvima	Single ingredient	5	Not controlled
Lorlatinib	Lorbrena	Single ingredient	3	Not controlled
Midostaurin	None listed	Single ingredient	1	Not controlled
Mirdametinib	Gomekli	Single ingredient	3	Not controlled
Momelotinib	Ojjaara	Single ingredient	3	Not controlled
Neratinib	Nerlynx	Single ingredient	1	Not controlled
Nilotinib	Tasigna, Danziten, Cavhanza	Single ingredient	25	Not controlled
Nintedanib esylate	Ofev	Single ingredient	24	Not controlled
Osimertinib	Tagrisso	Single ingredient	4	Not controlled
Pacritinib	Vonjo	Single ingredient	1	Not controlled
Palbociclib	Ibrance	Single ingredient	9	Not controlled
Pazopanib	Votrient	Single ingredient	9	Not controlled
Pemigatinib	Pemazyre	Single ingredient	3	Not controlled
Pexidartinib	Turalio	Single ingredient	1	Not controlled
Pirtobrutinib	Jaypirca	Single ingredient	2	Not controlled
Ponatinib	Iclusig	Single ingredient	4	Not controlled
Pralsetinib	Gavreto	Single ingredient	1	Not controlled
Quizartinib	Vanflyta	Single ingredient	2	Not controlled
Regorafenib	Stivarga	Single ingredient	1	Not controlled
Remibrutinib	Rhapsido	Single ingredient	1	Not controlled
Repotrectinib	Augtyro	Single ingredient	2	Not controlled
Ribociclib	Kisqali	Single ingredient	3	Not controlled
Ripretinib	Qinlock	Single ingredient	1	Not controlled
Ritlecitinib	Litfulo	Single ingredient	2	Not controlled
Ruxolitinib	Jakafi, Opzelura, Jakafi XR	Single ingredient	11	Not controlled
Selpercatinib	Retevmo	Single ingredient	6	Not controlled
Selumetinib	Koselugo	Single ingredient	4	Not controlled
Sirolimus	Hyftor, Fyarro	Single ingredient	39	Not controlled
Sorafenib	Nexavar	Single ingredient	9	Not controlled
Sunitinib malate	Sutent	Single ingredient	36	Not controlled
Taletrectinib adipate	Ibtrozi	Single ingredient	1	Not controlled
Tepotinib	Tepmetko	Single ingredient	1	Not controlled
Tivozanib	Fotivda	Single ingredient	2	Not controlled
Tovorafenib	Ojemda	Single ingredient	1	Not controlled
Trametinib dimethyl sulfoxide	Mekinist	Single ingredient	3	Not controlled
Trilaciclib	Cosela	Single ingredient	2	Not controlled
Tucatinib	Tukysa	Single ingredient	2	Not controlled
Vandetanib	Caprelsa	Single ingredient	2	Not controlled
Vemurafenib	Zelboraf	Single ingredient	1	Not controlled
Vimseltinib	Romvimza	Single ingredient	3	Not controlled
Zanubrutinib	Brukinsa	Single ingredient	2	Not controlled
Zongertinib	Hernexeos	Single ingredient	1	Not controlled

FDA established pharmacologic class: Kinase Inhibitor [EPC].

Questions

What drugs are Kinase Inhibitors?

The FDA NDC directory lists 71 single-ingredient drugs in this class: abemaciclib, acalabrutinib, afatinib, alectinib, avapritinib, axitinib, bosutinib, brigatinib, and more.

Where does this list come from?

From the established pharmacologic class (EPC) field FDA publishes for each listing in the NDC directory. A drug is listed when most of its prescription listings carry the class.

Kinase Inhibitors list

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Kinase Inhibitors (71)

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